Professional Documents
Culture Documents
Nucleic Essential
Membrane Protein
Cell wall acid metabolites
integrity synthesis
synthesis synthesis
Polype- Glyco-
B-lactam
ptides peptide -Nalidixic Quino- Sulfa Anti-
drugs Colistin Anti-
drugs drugs Amino Tetra- Chloroam- Macro- Linco- Fusidic acid Rifamycin lones drugs Tuber
(plymixen Fungal
glycosides cycline phenicol lides semides acid -Nitro Rifampin Fluro- (sulfona- culosis
E) Drugs
furantion quinoloes mides) drugs
Penicillins -Ex:INH+streptomycin
-Ketoconazole(oral)
imidazole Ethambutol+rifampin
-Clotrimazole(all
forms)
-Fluconazlo/Itraconazloe
Cephalo -New/more effective/less toxic
triazloe
sporins
-oral/topical for systematic
infections
Carba-
penems
polyenes Large circular molecule consisting
of hydrophilic & hydrophobic
regions
-Skin/hair infections
Mono-
Nystatin -Oral/topical
bactams
-safe
Ampho-
Tercin -systematic infections
B
-IV mainly
-Toxic
Cell wall
-Bacetracin
Vancomysin
Penicillins Cephalosporins Carbapenems monobactams -Colistin
Teicoplanin
(polymixen B)
-Bactericidal
-Affect + Anaerobic/narrow
spec. *A* *B* *C* *D*
Methicillin
Oxacillin Cloxacillin Augmentin
-applied topically
Erythromycin
Doxycycline (creams/eye drops)
Tuberculosis streptomycin minocycline
Clarithromycin
-for skin infections
azithromycin
-steroidal/prevent
t-RNA translocation
To ribosomes
-Broad spectrum. -For UT/RT infections like -not used in system.
-Orally or injected Pneumonia & diphtheria Infections very toxic
Neomycin (orally more common) -For mycoplasma/clamydia/ -metronidazol(flagyl)
Intestinal infection Konamycin -Not given to cildren Staphylococcus/legionella is an example.
Under 8 Infections
-For Ut/Rt infections -inhibit peptidyl
Caused by transferase activity
mycoplasma & translocation
Meningitis Gentamycin ,clamydia and of growing peptide to
Tobramycin Legionella. Ribosome
sepsis Netilimycin -most applied orally/less IV
Amikacin
-prevent transcription
-affect mainly G-Ve
by binding to RNA Norfloxacin UT/RT infections
Bacteria in
Polymerase
UT.
-Broad spectrum
-for UT infections
-effective in killing
-used agains E.coli (responsible UT/RT(pneumonia)/
IC Bacteria
For 70%-80% of UT Intestinal/blood
-used for serious infection Ciprofloxacin
Infections) (septicemia)
Meningitis /brucellosis
-Acts on DNA gyrase infections
Not for simple RT infection
(type of DNA
(WHO)
Polymerase)
-Bacteria May produce enzyme
affect B Subunits in RNA Levofloxacin
Polymerase Developing
Upper RT infections
resistance to these drugs
-less toxic then aminoglysocides.