Shiela Mae S. Torres 2BMT CHOLINOCEPTOR-ACTIVATING & CHOLINESTERASE-INHIBITING DRUGS I. Direct Acting (Receptor Agonist) 1. Muscarinic a.

Choline esters 1. Acetylcholine a. Miochol-E b. Miochol-E/Steri-Tags c. Miochol 2. Metacholine a. Provocholine b. c. 3. Bethanechol a. Urecholine b. Duvoid c. Myotonachol 4. Carbachol a. Miostat b. Carboptic c. Isopto Carbachol b. Alkaloids 1. Muscarine a. b. c. 2. Pilocarpine a. Salagen b. Akarpine c. Almocarpine 2. Nicotinic a. Ganglionic 1. Nicotine a. Nicoderm CQ b. Nicorette c. Nicotrol Inhaler 2. Lobeline a. Lobeline Harvest Pharm b. Zoolobelin (veterinary use) c. Smokeless 3. DMPP (dimethylphenylpiperazinium) a.

Shiela Mae S. Torres 2BMT b. c. 4. Varenicline a. Chantix b. Champix c. b. Neuromuscular 1. Nicotine a. Nic-Sal b. Nico-Dust c. Nico-Fume II. Indirect-Acting (Cholinesterase Inhibitors) 1. Reversible a. Edrophonium 1. Antirex 2. Enlon 3. Enlon Plus b. Carbamates 1. Neostigmine a. Prostigmin Bromide b. Neostigmine omega c. Prostigmin 2. Physostigmine a. Antilirium b. Esromiotin c. Ezerin 3. Pyridostigmine a. Mestinon b. Mestinon-SR c. Regonol 4. Demacarium a. Humorsol Ocumeter b. c. 5. Ambenonium a. Mytelase Chloride b. Mytelase c. 2. Irreversible a. Phosphates 1. Echothiopate

Shiela Mae S. Torres 2BMT a. Echodide b. Phospholine Iodide (Wyeth-Ayerst) c. Isoflurophate a. Dyflos b. Floropryl c. Fluorodiisopropyl Phosphate Soman (nerve gas) a. b. c. Parathion a. b. c. Malathion a. Lice Rid b. Malacide c. Malafor Sarin a. b.

2.

3.

4.

5.

6.

CHOLINOCEPTOR BLOCKING DRUGS I. Muscarinic Antagonists 1. Belladonna Alkaloids a. Atropine 1. Atrosulf 2. Equipin 3. Eyesules b. Scopolamine 1. Euscopol 2. Hydroscine Hydrobromide 3. Hyocine F Hydrobromide 2. Synthetic Tertiary Amines a. Pirenzepine 1. Bisvanil 2. Gasteril 3. Gastrozepin b. Dicyclomine 1. Atumin

Shiela Mae S. Torres 2BMT 2. Bentomine 3. Bentyl c. Tropicamine 1. Mydriacyl 2. Mydriafair 3. Mydriaticum 3. Quaternary Amines a. Glycopyrrolate 1. Asecryl 2. Gastrodyn 3. Nodapton b. Homatropine 1. Novatrin 2. Novatrine 3. Novatropine c. Propantheline 1. Pro-Banthine 2. Propanthel 3. d. Ipratropium 1. Apovent 2. Atronase 3. Atrovent e. Benztropine 1. Akitan 2. Apo-Benztropine (Apotex) 3. Cobrentin II. Nicotinic Antagonists 1. Ganglionic Blockers a. Tetraethylammonium (TEA) 1. 2. 3. b. Hexamethonium 1. 2. 3. c. Decamethonium 1. Lopac-D-1260 2. Syncurine 3.

Shiela Mae S. Torres 2BMT d. Mecamylamine 1. Inversine 2. Inversine hydrochloride 3. Mecamine e. Trimethapan 1. Arfonad 2. 3. 2. Neuromuscular Blockers a. Nondepolarizing 1. Tubocurarine a. Curare b. Delacurarine c. Jexin 2. Pancuronium a. Mioblock b. Pavulon c. 3. Atracurium a. b. c. 4. Vecuronium a. b. c. b. Depolarizing 1. Succinylcholine a. Anectine b. Quelicin c. Quelicin Preservative Free

Shiela Mae S. Torres 2BMT