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PROTEIN INHIBITORS
* BROAD-SPECTRUM ANTIBIOTIC
1. TETRACYCLINE
-uses: resistant to almost ALL gram +/- COCCI except for N.gonorrhea but
sensitive to bacilli
-class:
-pk:
iii. x in csf
2. CHLORAMPHENICOL
-moa: inhibit bact protein synthesis (50S), - 70S causes host toxicity
-pk:
i. oral
iii. liverurine
-class:
i. natural- erythromycin
-pk:
i. x in csf
ii. liverbile
4. CLINDAMYCIN
5. LINEZOLID
-general: synthetic,bacteriostatic
6. KETOLIDES
Lect 2
* BROAD-SPECTRUM ANTIBIOTICS
* BACTERICIDAL
BETA-LACTAMS
1. PENICILLINS
-class:
ii. semisynthetic-
a. AMPICILLIN (sulbactam)
PIPERACILLIN (tazobactam)
-class:
ii. 2nd
iii. 3rd
3. CARBAPENEM
-progrug: imipenem
-pk: only iv
4. MONOBACTAM
-prodrug: aztreonam
Lect 3
AMINOGLYCOSIDES
-prodrugs:
i. streptomycin
ii. gentamycin
iii. amikacin
iv. neomycin
- BACTERICIDAL
-pk:
ii. x in csf
Lect 4
SPECTINOMYCIN
- bacteriostatic
-a/e: hypersensitivity
Lect 5
1. SULPHONAMIDES
i. oral
a. sulfadiazine – short
c. sulfadoxine – long
-pk:
i. NEVER given iv or im
iii. liverurine
2. TRIMETHOPRIM
-pk:
i. oral
-iv or oral